Table 8 The characterization of the F2 peptide as an inhibitor of the GST-catalyzed reaction (The Vmax, Ki and [I]/Ki values of the GST-catalyzed reaction in the presence of the F2 inhibit peptide were determined).
From: A novel method for screening the glutathione transferase inhibitors
F2 peptide concentration [I] (μM) | Km value (mM) | Ki value (μM) | [I]/Ki |
|---|---|---|---|
0 | 0.25 | - | - |
0.8 | 0.38 | 1.53 | 0.52 |
1.6 | 0.50 | 1.60 | 1.0 |
3.2 | 0.58 | 2.42 | 1.32 |