Pex5p(C): | Ligand | n | ΔH (kJ/mol) | TΔS (kJ/mol) | ΔG (kJ/mol) | Kd (nM) |
---|---|---|---|---|---|---|
Wild-type (5) a | mSCP2 | 0.93 ± 0.03 | -43.4 | -1.8 | -42.3 | 95 ± 21 |
R608W (4) | mSCP2 | 0.61 ± 0.06 | -71.7 | -31.8 | -39.9 | 179 ± 19 |
D624W (4) | mSCP2 | 0.41 ± 0.08 | -55.6 | -12.2 | -43.4 | 45 ± 8 |
Wild-type (2) | PGNAKL | 0.94 ± 0.02 | -42.5 | -5.6 | -36.9 | 547 ± 6 |
R608W (2) | PGNAKL | 0.81 ± 0.01 | -51.6 | -15.1 | -36.5 | 635 ± 25 |
D624W (2) | PGNAKL | 0.49 ± 0.01 | -54.7 | -18.6 | -36.1 | 763 ± 0 |