Table 7 The characterization of the F1 peptide as an inhibitor of the GST-catalyzed reaction (The Vmax, Ki and [I]/Ki values of the GST-catalyzed reaction in the presence of the F1 inhibit peptide were determined).
From: A novel method for screening the glutathione transferase inhibitors
F1 peptide concentration [I] (μM) | Vmax value (μmol/mg/min) | Ki value (μM) | [I]/Ki |
|---|---|---|---|
0 | 1.0 | - | - |
0.8 | 0.833 | 4.0 | 0.2 |
1.6 | 0.741 | 4.57 | 0.35 |
3.2 | 0.645 | 5.82 | 0.55 |